5-Iodo-A-85380 dihydrochloride - CAS 1217837-17-6
Category: Inhibitor
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Molecular Formula:
C9H13IN2OCl2
Molecular Weight:
363.03
COA:
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Targets:
nAChR
Description:
5-Iodo-A-85380 dihydrochloride is the dihydrochloride salt of 5-Iodo-A-85380, which is a highly potent and subtype-selective agonist for α4β2 and α6β2 nicotinic acetylcholine receptors. It activates α-CTx-MII-sensitive and -insensitive components of [3H]dopamine release from rat striatal synaptosomes.
Purity:
≥99% by HPLC
Synonyms:
3-[(2S)-2-Azetidinylmethoxy]-5-iodopyridine dihydrochloride
MSDS:
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InChIKey:
ZJVVFYWEBSHGBV-JZGIKJSDSA-N
InChI:
InChI=1S/C9H11IN2O.2ClH/c10-7-3-9(5-11-4-7)13-6-8-1-2-12-8;;/h3-5,8,12H,1-2,6H2;2*1H/t8-;;/m0../s1
Canonical SMILES:
C1CNC1COC2=CC(=CN=C2)I.Cl.Cl
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CAS 1217837-17-6 5-Iodo-A-85380 dihydrochloride

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