|Description||(±)-5'-Chloro-5'-deoxy-ENBA is a selective adenosine A1 receptor agonist (Ki = 0.51, 1290, 1340 and 2740 nM at A1, A3, A2A and A2B receptors respectively). It is used as an antinociceptive.|
|Brife Description||adenosine A1 receptor agonist|
|Purity||≥98% by HPLC|
SLV 320 is a potent and selective adenosine A1 receptor antagonist (Ki = 1, 200, 398 and 3981 nM at human A1, A3, A2A and A2B receptors, respectively). SLV320 p...
UP202-56, an adenosine analogue, selectively acts via A1 receptors to significantly decrease noxiously-evoked spinal c-Fos protein expression.
PSB 11 hydrochloride
PSB 11 hydrochloride, an anti-inflammatory imidazopurinone, has displayed potent and highly selective antagonist characteristics towards human Adenosine A3-R, w...
GR 79236, an effective Adenosine A1 receptor agonist, could probably be used as an anti-inflammatory agent. IC50: 3.1 nM(Ki).
CGH 2466 dihydrochloride
CGH 2466 dihydrochloride is an adenosine A1, A2B and A3 receptor antagonist (IC50 = 19, 21, and 80 nM, respectively). It also displays an inhibitory effect on p...
CVT5440 is a selective, high affinity A(2B) adenosine receptor antagonist. It may has the potential treatment of asthma and has good selectivity.
8-Aminoadenine is an adenine receptor agonist with Ki value of 0.0341 μM in HEK293 cells expressing an adenine binding site. It shows 190-fold increased potency...
Naxifylline, a xanthine derivative, has been found to be an adenosine A1 receptor antagonist as well as diuretic agent that was once studied in heart failure an...