|Description||(-)-[3R,4S]-Chromanol 293B is one of the chromanols, which inhibits cAMP-mediated Cl- secretion in colon crypts by a blockade of a cAMP-activated K+ conductance. It selectively inhibits the slow component of delayed rectifier K+ current. It has negligible inhibitory action at KV11.1 (hERG) channels. It may be a useful research chemical.|
|Purity||≥99% by HPLC|
Pipemidic acid is a synthetic quinolone antibiotic agent as a ATP-sensitive K+ channel blocker.
PNU 37883 hydrochloride
PNU 37883 is a potent, euglycemic vascular K-ATP blocker that also exerts a K+-sparing diuresis at higher doses. It selectively inhibits Kir6 currents in isolat...
NS5806 is a KV4.3 channel activator. It can mediate the transient outward K+ current (Ito).
Tertiapin-Q, a derivative of the bee venom toxin tertiapin, is a high affinity blocker of inward-rectifier K+ channels. Tertiapin-Q binds to ROMK1 (Kir1.1) and ...
AZD1305 is a potassium channel and sodium channel antagonist. It can inhibit rapidly the activating delayed-rectifier potassium current, L-type calcium current,...
DMP 543 is an acetylcholine release stimulator and a K-ATP channel blocker. It significantly enhances K+-stimulated [3H]-ACh release from rat hippocampal slices...
Psora 4 is the most potent small-molecule Kv1.3 blocker known. It blocked Kv1.3 in a use-dependent manner, with a Hill coefficient of 2 and an EC50value of 3 nM...
Mitiglinide calcium hydrate
Mitiglinide calcium hydrate, a derivative of benzylsuccinic acid, is a highly selective K-ATP channel antagonist.