3-MPPI - CAS 133399-65-2
Category: Inhibitor
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Molecular Formula:
C23H25N5O3
Molecular Weight:
419.48
COA:
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Targets:
Adrenergic Receptor
Description:
3-MPPI is a very potent ligand for α1 sites (Ki for displacement of prazosin = 0.2 nM) and regulates smooth muscle contraction. 3-MPPI shows different binding properties for each α1 subtype (pKi values are 8.74, 9.44 and 9.57 for α1B, α1D and α1A adrenoceptors respectively).
Synonyms:
2-[(4-Phenylpiperazin-1-yl)methyl]-2,3-dihydroimidazo[1,2-c]quinazolin-5(6H)-one
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
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InChIKey:
AQASGOHUMGAWJJ-UHFFFAOYSA-N
InChI:
InChI=1S/C23H25N5O3/c1-31-19-9-5-4-8-18(19)27-13-10-26(11-14-27)12-15-28-22(29)21-20(25-23(28)30)16-6-2-3-7-17(16)24-21/h2-9,24H,10-15H2,1H3,(H,25,30)
Canonical SMILES:
COC1=CC=CC=C1N2CCN(CC2)CCN3C(=O)C4=C(C5=CC=CC=C5N4)NC3=O
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CAS 133399-65-2 3-MPPI

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