(1R,2S)-VU0155041 - CAS 1263273-14-8
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C14H15Cl2NO3
Molecular Weight:
316.18
COA:
Inquire
Targets:
mGluR
Description:
(1R,2S)-VU0155041 is a partial mGluR4-positive allosteric modulator (EC50= 2.35 μM) that dependently attenuated hyperalgesia in neuropathic pain model rats.
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Brife Description:
A partial mGluR4 agonist (EC50= 2.35 μM)
Synonyms:
(1R,2S)-2-[(3,5-dichlorophenyl)carbamoyl]cyclohexane-1-carboxylic acid; VU 0155041; VU-0155041; VU0155041
Solubility:
DMSO: ≥ 59 mg/mL
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
540.2±50.0 ℃ at 760 Torr
Density:
1.429±0.06 g/cm3
InChIKey:
VSMUYYFJVFSVCA-NWDGAFQWSA-N
InChI:
1S/C14H15Cl2NO3/c15-8-5-9(16)7-10(6-8)17-13(18)11-3-1-2-4-12(11)14(19)20/h5-7,11-12H,1-4H2,(H,17,18)(H,19,20)/t11-,12+/m0/s1
Canonical SMILES:
C1CCC(C(C1)C(=O)NC2=CC(=CC(=C2)Cl)Cl)C(=O)O
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CAS 1263273-14-8 (1R,2S)-VU0155041

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