(R)-6-Hydroxybuspirone hydrochloride - CAS 477930-30-6
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
(R)-6-Hydroxybuspirone hydrochloride
Catalog Number:
477930-30-6
Synonyms:
6-hydroxy-8-(4-(4-(2-pyrimidinyl)-1-piperazinyl)butyl)-, (6R)-8-Azaspiro(4.5)decane-7,9-dione
CAS Number:
477930-30-6
Description:
(R)-6-Hydroxybuspirone is a major active metabolite of Buspirone. (R)-Enantiomer showed higher affinity and selectivity for the 5HT1A receptor compared to the (S)-enantiomer; while (S)-Enantiomer has advantage of being cleared more slowly from blood compared to the (R)-enantiomer
Molecular Weight:
401.5
Molecular Formula:
C21H31N5O3
Quantity:
Milligrams-Grams
Quality Standard:
Enterprise standard
COA:
Inquire
MSDS:
Inquire
Canonical SMILES:
c1cnc(nc1)N2CCN(CC2)CCCCN3C(=O)CC4(CCCC4)[C@H](C3=O)O
InChI:
1S/C21H31N5O3/c27-17-16-21(6-1-2-7-21)18(28)19(29)26(17)11-4-3-10-24-12-14-25(15-13-24)20-22-8-5-9-23-20/h5,8-9,18,28H,1-4,6-7,10-16H2/t18-/m0/s1
InChIKey:
KOZNAHJIJGCFJJ-SFHVURJKSA-N
Targets:
5-HT Receptor
Current Developer:
Bristol-Myers Squibb

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