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KRP297 - CAS 213252-19-8

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Category
Inhibitor
Product Name
KRP297
Catalog Number
213252-19-8
Synonyms
5-[(2,4-dioxo-1,3-thiazolidin-5-yl)methyl]-2-methoxy-N-[[4-(trifluoromethyl)phenyl]methyl]benzamide; KCL1998001079; KRP 297; KRP-297; KRP297; L 410198; L-410198; L410198; MK 767; MK-767
CAS Number
213252-19-8
Description
KRP297, also called as L4 10198 or MK 767, is a Peroxisome proliferator-activated receptor (PPAR) alpha and gamma (PPARα and PPARγ) agonist. With potential to treat type 2 diabetes and dyslipidemia, KRP297 is able to decrease plasma glucose and insulin levels.
Molecular Weight
438.42
Molecular Formula
C20H17F3N2O4S
COA
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MSDS
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Canonical SMILES
COC1=C(C=C(C=C1)CC2C(=O)NC(=O)S2)C(=O)NCC3=CC=C(C=C3)C(F)(F)F
InChI
1S/C20H17F3N2O4S/c1-29-15-7-4-12(9-16-18(27)25-19(28)30-16)8-14(15)17(26)24-10-11-2-5-13(6-3-11)20(21,22)23/h2-8,16H,9-10H2,1H3,(H,24,26)(H,25,27,28)
InChIKey
NFFXEUUOMTXWCX-UHFFFAOYSA-N
Targets
PPAR
Structure
CAS 213252-19-8 KRP297
Specification
Purity
>98%
Appearance
Solid powder
Solubility
Soluble in DMSO
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