Nitrodienamine, an inhibitor of Ca2+/Mg2+ ATPase.
Quinoline alkaloid, extracted from Haplophyllum bucharicum (Rutacae)
Diterpenoid , from plants of the Stevia genus, Compositae. Sweetener; reported as possessing anti-hypertensive effects upon hypertensive rats.
A SR-4 agonist with moderate activity as a SR-3 antagonist
Ducamycin Analog is a cytotoxic agent, used as the cytotoxic component in antibody-drug conjugates.
A Norditerpenoid alkaloid. Nicotinic receptor antagonist at the neuromuscular junction and vegetative ganglia; hypotensive. Diterpene alkaloid , from plants of ...
An antiarrhythmic of 1-st and 1Y classes and a blocker of TTX sensitive Na+ channels, Ca++ antagonist diterpene alkaloid from Delphinium staphisagria.
ω-agatoxin-IVA (ω-AGA IVA) is a peptide originally isolated from funnel web-spider venom Agelenopsis aperta. This peptide is a specific blocker of P/Q-type calc...
Tetrahydroberberine is a protoberberine alkaloid which potently block functional KATP channels natively expressed on midbrain dopamine neurons. Tetrahydroberber...
C20-diterpenoid alkaloid , from the Ranunculaceae family,an antiarrhythmic.
Daun02 is a daunorubicin b-galactoside prodrug for use in conjunction.
Lignan , from plants of the Rutaceae family, a substance presenting an estrogenic activity and sedative effects. .
A selective inhibitor of endoplasmic reticulum Ca2+-ATPase.
α-conotoxin GI (alpha-conotoxin GI) is a conopeptide that has been isolated from the venom of the cone snail Conus geographus. α-conotoxin GI is a competitive a...
Synthetic, an inhibitor of high-affinity choline uptake (HAChU) in synaptosomes.
Potent inhibitor of protein phosphatase tyoe 1 (PP1) and protein phosphatase tyoe 2A (PP2A).
Synthetic, GABAA-gated Cl- channels blocker; non-competitive GABAA antagonist.
Potent blocker of voltage-sensitive K+ channels (IC50 values are 0.1, 1.1 and 25 nM for KV1.3, KV1.1 and KV1.2 channels) respectively). Also inhibits Ca2+-activ...
Used as an antihypertensive and antianginal. A dihydorpyridine calcium channel blocker.
Melittin inhibits protein kinase C, Ca2+/calmodulin-dependent protein kinase II, myosin light chain kinase and Na+/K+-ATPase (synaptosomal membrane) and is a ce...