(+)-Apogossypol - CAS 66389-74-0
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
(+)-Apogossypol
Catalog Number:
66389-74-0
Synonyms:
(R)-5,5'-diisopropyl-3,3'-dimethyl-[2,2'-binaphthalene]-1,1',6,6',7,7'-hexaol; methanol;3-methyl-5-propan-2-yl-2-(1,6,7-trihydroxy-3-methyl-5-propan-2-ylnaphthalen-2-yl)naphthalene-1,6,7-triol; Apogossypol;
CAS Number:
66389-74-0
Description:
(+)-Apogossypol is a potent inhibitor of Bcl-2 family proteins, binding and inhibiting Bcl-2 and Bcl-X(L) with high affinity and induces apoptosis of tumor cell lines.
Molecular Weight:
494.58
Molecular Formula:
C29H34O7
Quantity:
Milligrams-Grams
Quality Standard:
Enterprise Standard
COA:
Inquire
MSDS:
Inquire
Canonical SMILES:
CC1=C(C(=C2C=C(C(=C(C2=C1)C(C)C)O)O)O)C3=C(C=C4C(=C3O)C=C(C(=C4C(C)C)O)O)C.CO
InChI:
1S/C28H30O6.CH4O/c1-11(2)21-15-7-13(5)23(25(31)17(15)9-19(29)27(21)33)24-14(6)8-16-18(26(24)32)10-20(30)28(34)22(16)12(3)4;1-2/h7-12,29-34H,1-6H3;2H,1H3
InChIKey:
DDVSMQNLYHXDSK-UHFFFAOYSA-N
Targets:
Bcl-2 Family
Current Developer:
Coronado Biosciences

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