Alvimopan - CAS 156053-89-3
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
Alvimopan
Catalog Number:
156053-89-3
Synonyms:
2-[[(2S)-2-benzyl-3-[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl]propanoyl]amino]acetic acid ADL 8-2698 ADL8-2698 alvimopan alvimopan anhydrous anhydrous alvimopan Entereg LY 246736 LY-246736 LY246736 trans-3,4-dimethyl-4-(3-hydroxyphenyl) pipe
CAS Number:
156053-89-3
Description:
Alvimopan is a novel, oral, peripherally acting antagonist of the mu opioid receptor, which can help gastrointestinal recovery after surgery. Phase III IC50: Mu-type opioid receptor= 1.7 nM
Molecular Weight:
424.53
Molecular Formula:
C25H32N2O4
Quantity:
Grams-Kilos
COA:
Inquire
MSDS:
Inquire
Canonical SMILES:
CC1CN(CCC1(C)C2=CC(=CC=C2)O)CC(CC3=CC=CC=C3)C(=O)NCC(=O)O
InChI:
1S/C25H32N2O4/c1-18-16-27(12-11-25(18,2)21-9-6-10-22(28)14-21)17-20(24(31)26-15-23(29)30)13-19-7-4-3-5-8-19/h3-10,14,18,20,28H,11-13,15-17H2,1-2H3,(H,26,31)(H,29,30)/t18-,20-,25+/m0/s1
InChIKey:
UPNUIXSCZBYVBB-JVFUWBCBSA-N
Targets:
Opioid Receptor
Current Developer:
Adolor Corporation; Cubist Pharmaceuticals
Chemical Structure
CAS 156053-89-3 Alvimopan

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