AL 082D06 - CAS 256925-03-8
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
AL 082D06
Catalog Number:
256925-03-8
Synonyms:
1S/C23H24ClN3O2/c1-25(2)18-9-5-16(6-10-18)23(17-7-11-19(12-8-17)26(3)4)21-15-20(27(28)29)13-14-22(21)24/h5-15,23H,1-4H3 IPICUXHYPAMJNC-UHFFFAOYSA-N CN(C)C1=CC=C(C=C1)C(C2=CC=C(C=C2)N(C)C)C3=C(C=CC(=C3)[N+](=O)[O-])Cl
CAS Number:
256925-03-8
Description:
AL 082D06, also called as D-06, is a selective nonsteroidal antagonist of glucocorticoid receptor (GR) (Ki= 210 nM) without significant activity on AR, PR, MR and ER(Ki > 10 uM). AL 082D06 binds competitively with steroids, likely occupying a similar site
Molecular Weight:
409.91
Molecular Formula:
C23H24ClN3O2
COA:
Inquire
MSDS:
Inquire
Canonical SMILES:
CN(C)C1=CC=C(C=C1)C(C2=CC=C(C=C2)N(C)C)C3=C(C=CC(=C3)[N+](=O)[O-])Cl
InChI:
1S/C23H24ClN3O2/c1-25(2)18-9-5-16(6-10-18)23(17-7-11-19(12-8-17)26(3)4)21-15-20(27(28)29)13-14-22(21)24/h5-15,23H,1-4H3
InChIKey:
IPICUXHYPAMJNC-UHFFFAOYSA-N
Targets:
Glucocorticoid Receptor

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