AGN 196996 - CAS 958295-17-5
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
AGN 196996
Catalog Number:
958295-17-5
CAS Number:
958295-17-5
Description:
AGN 196996 is a potent and selective antagonist of RARα. It has been reported to selectively bind to RARs (retinoic acid receptors) for RARα, RARβ and RARγ. It can inhibit the gene transcription activity which induced by ATRA and other RAR agonists. It shows no activity in transactivation assays, but instead block the gene transcriptional activity induced by ATRA and other RAR agonists.
Molecular Weight:
482.32
Molecular Formula:
C24H20BrNO5
COA:
Inquire
MSDS:
Inquire
Targets:
RAR/RXR
Chemical Structure
CAS 958295-17-5 AGN 196996

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