|Description||This active molecular is a reversible and selective platelet P2Y12 receptor antagonist. IC50 value of ACT-246475 is 8.0 nM. ACT-246475 dose-dependently blocked thrombus formation in the rat ferric chloride model and displayed a wide therapeutic window. In May 2016, Phase-I development is ongoing in France.|
|Quality Standard||In-house standard|
|Current Developer||Originator:Actelion Pharmaceuticals|
Riboflavin phosphate sodium
Riboflavin phosphate sodium, a Riboflavin derivative, is a commonly existed nutritional factor and could improve the biomechanical stiffness of corneal.
Erythromycin Ethylsuccinate, an oral macrolide antibiotic produced by Streptomyces erythreus, reversibly binds to the 50S ribosome of bacteria, and inhibits pro...
Ro 48-8071 fumarate
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Aminocaproic acid is a derivative and analogue of the amino acid lysine, which makes it an effective inhibitor for enzymes that bind that particular residue. Su...
Benflumetol, also known as HSDB 7210, is an antimalarial drug used to treat acute uncomplicated malaria. It is used in combination with Artemether for improved ...
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Clofentezine is an active substance of plant protection product used as pesticide, acaricide. It belongs to the chemical family of quinoxalines. It is used in a...
Aluminum phthalocyanine tetrasulfonate t
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Clonidine is an α2-Adrenergic agonist for neuropathic pain.
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trans-Tetrahydro-4-methylene-2-octyl-5-oxo-3-furancarboxylic Acid is a well-known fatty acid synthase (FAS) inhibitor. Studies show that trans-Tetrahydro-4-meth...
Aloin B is one isomer of Aloin; Aloin is a physiologically active anthraquinone present in aloe.