aceprometazine - CAS 13461-01-3
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
aceprometazine
Catalog Number:
13461-01-3
Synonyms:
aceprometazine;1-[10-[2-(Dimethylamino)propyl]-10H-phenothiazin-2-yl]ethanone;Acepromethazine
CAS Number:
13461-01-3
Description:
Aceprometazine is a Histamine H1 receptor antagonist as an approved drug. It can be used in combination with meprobamate for the treatment of sleep disorders such as Insomnia.
Molecular Weight:
326.46
Molecular Formula:
C19H22N2OS
Quantity:
Milligrams-Grams
Quality Standard:
In-house standard
COA:
Inquire
MSDS:
Inquire
Canonical SMILES:
CC(CN1C2=CC=CC=C2SC3=C1C=C(C=C3)C(=O)C)N(C)C
InChI:
InChI=1S/C19H22N2OS/c1-13(20(3)4)12-21-16-7-5-6-8-18(16)23-19-10-9-15(14(2)22)11-17(19)21/h5-11,13H,12H2,1-4H3
InChIKey:
XLOQNFNTQIRSOX-UHFFFAOYSA-N
Targets:
Histamine Receptor
Chemical Structure
CAS 13461-01-3 aceprometazine

Related Histamine Receptor Products


CAS 140462-76-6 Olopatadine HCl

Olopatadine HCl
(CAS: 140462-76-6)

Olopatadine HCl is a histamine blocker and mast cell stabilizer with an IC50 of 559 μM for the release of histamine

CAS 1229-35-2 METHDILAZINE HYDROCHLORIDE (200 MG)

METHDILAZINE HYDROCHLORIDE (200 MG)
(CAS: 1229-35-2)

This active molecular is a first-generation antihistamine and belongs to phenothiazine class. Methdilazine Hydrochloride is a Histamine H1 receptor antagonist w...

CAS 13461-01-3 aceprometazine

aceprometazine
(CAS: 13461-01-3)

Aceprometazine is a Histamine H1 receptor antagonist as an approved drug. It can be used in combination with meprobamate for the treatment of sleep disorders su...

CAS 113-92-8 Chlorpheniramine Maleate

Chlorpheniramine Maleate
(CAS: 113-92-8)

Chlorpheniramine inhibits the proliferation of MCF-7, MDA-MB 231, and Ehrlich cells in a dose-response manner, and significantly reduces the ornithine decarboxy...

CAS 903576-44-3 BF 2649

BF 2649
(CAS: 903576-44-3)

Pitolisant hydrochloride is an antagonist of the histamine H3 receptor, which is used for the treatment of narcolepsy with or without cataplexy in adult patient...

CAS 202189-78-4 Bilastine

Bilastine
(CAS: 202189-78-4)

Bilastine is a novel, nonsedating H1-antihistamine developed for symptomatic treatment of allergic rhinitis and chronic idiopathic urticaria.

CAS 10246-75-0 Hydroxyzine pamoate

Hydroxyzine pamoate
(CAS: 10246-75-0)

Hydroxyzine pamoate, a derivative of hydroxyzine, is a histamine H1-receptor antagonist that has been used as anxiolytic and antihistaminic so that it is probab...

CAS 132-20-7 Pheniramine Maleate

Pheniramine Maleate
(CAS: 132-20-7)

Pheniramine Maleate is an antihistamine with anticholinergic properties used to treat allergic conditions such as hay fever or urticaria.

CAS 132-21-8 dexbrompheniramine

dexbrompheniramine
(CAS: 132-21-8)

Dexbrompheniramine is an histamine H1-receptor antagonist used for the treatment of allergic conditions including hay fever or urticaria. It is the pharmacologi...

CAS 59-33-6 Pyrilamine maleate salt

Pyrilamine maleate salt
(CAS: 59-33-6)

Pyrilamine maleate salt is a first generation antihistamine and binds with high affinity to G(q/11) protein. It is commonly utilized as a radioligand binding as...

CAS 544707-19-9 JNJ10181457 dihydrochloride

JNJ10181457 dihydrochloride
(CAS: 544707-19-9)

JNJ10181457 dihydrochloride is a selective non-imidazole brain penetrant histamine H3 receptor antagonist with pKi values of 8.15 and 8.93 for rat and human H3 ...

KDM5A-IN-1
(CAS: 1905481-36-8)

KDM5A-IN-1, a pyrrolidine amide compound, is an inhibitor histone demethylases.

CAS 442-52-4 Clemizole

Clemizole
(CAS: 442-52-4)

Clemizole is an H1 antagonist acts as a TRPC5 channel blocker (IC50 values are 1.1, 6.4, 9.1, 11.3 and 26.5 μM for TRPC5, TRPC4, TRPC3, TRPC6 and TRPC7 respecti...

UR-PI376
(CAS: 1192559-94-6)

This active molecular is a imidazolylpropylguanidine type compound as a hH4R agonist (histamine H4 receptor agonist) showing negligible hH1R and hH2R activities...

Levoprotiline hydrochloride
(CAS: 76496-69-0)

Levoprotiline is a Histamine H1 receptor antagonist originated by Novartis. It is an antidepressant. But clinical trials for Major depressive disorder were disc...

CAS 93793-83-0 Roxatidine Acetate HCl

Roxatidine Acetate HCl
(CAS: 93793-83-0)

Roxatidine Acetate HCl is a specific and competitive histamin H2 receptor antagonist.

CAS 77-38-3 Chlorphenoxamine

Chlorphenoxamine
(CAS: 77-38-3)

Chlorphenoxamine is an analog of diphenhydramine. It has antimuscarinic and antihistaminic properties. It has been used as an antipruritic and antiparkinsonian ...

CAS 153439-40-8 Fexofenadine HCl

Fexofenadine HCl
(CAS: 153439-40-8)

Fexofenadine inhibits histamine H1 receptor with IC50 of 246 nM.

Mizolastine dihydrochloride
(CAS: 1056596-82-7)

The dihydrochloride salt form of Mizolastine which is effective in the treatment of seasonal allergic rhinitis, perennial allergic rhinitis and other allergy sy...

CAS 34839-70-8 Metiamide

Metiamide
(CAS: 34839-70-8)

Metiamide is developed from another burimamide, used as a histamine H2 receptor antagonist.