|Synonyms||BAY g 5421|
|Description||Acarbose is an inhibitor of intestinal alpha-glucosidase, used to treat type 2 diabetes mellitus.|
CB 3703 is an inhibitor of hydrofolate reductase.
Ocaphane Hydrochloride is a strong antitumor agent used on a number of animal tumors such as Brown-Pearce carcinoma but is fairly toxic to hemopoietic organs.
MDL-72274 is a selective SSAO inhibitor. It is a potent (IC50 = 10(-9) M) inhibitor of both MAO-B and SSAO, with 190-fold lower affinity for MAO-A. MDL-72974 ca...
Endochin is an experimental antimalarial which was known to be causal prophylactic and potent erythrocytic stage agents in avian models.
L-NAME is a nonselective inhibitor of nitric oxide synthetases (NOS) for nNOS (bovine), eNOS (human), and iNOS (murine), with Ki of 15 nM, 39 nM and 4.4 μM, res...
Dronedarone is a Class III antiarrhythmic and a multi-channel blocker for atrial fibrillation. It blocks potassium, sodium, and calcium channels and also exhibi...
Dirlotapide is a drug used to treat obesity in dogs works as a gut-selective microsomal triglyceride transfer protein (MTTP or MTP) inhibitor.
Vapreotide is a synthetic somatostatin analog as a Somatotropin receptor antagonist. It can be used for the treatment of esophageal variceal bleeding in patient...
Pocapavir has been found to be an antienterovirus agent that could probably be effctive against enterovirus infections. The Phase-II trial for Poliomyelitis has...
JZP-430, a thiadiazol derivative, has been found to be an ABHD6 inhibitor that could probably be effective in obesity and type II diabetes therapy. IC50: 44 nM.
FR 121196 is a potential antidementia drug originated by Fujisawa. Mechanism of Action is not undefined. FR 121196 can ameliorate the impaired memory of rat in ...
Mebeverine Acid is a metabolite of Mebeverine, an antispasmodic. Mebeverine acid appears to be a valuable marker of oral exposure to Mebeverine.
Tirapazamine is a benzotriazine di-N-oxide with potential antineoplastic activity. Tirapazamine is selectively activated by multiple reductases to form free rad...
Octocrylene is an organic compound used as an ingredient in sunscreens and cosmetics.
Halobetasol propionate act by the induction of phospholipase A2 inhibitory proteins.
Ginsenoside Rg3 is a natural product isolated from Panax ginseng. Similar to other ginsenosides it exhibits cardio protective effects. Ginsenoside Rg3 enhances ...
Tofisopam, a 2,3-benzodiazepine, has depressant effects at high doses in several different animal test procedures. Tofisopam has been shown to enhance the antic...
D-Luciferin sodium salt
Sodium salt form of D-Luciferin, derived from the luciferase gene of photinus pyralis, is commonly used as a reporter gene for studying transcriptional regulati...
JPH203 is a potent and selective L-type amino acid transporter 1 (LAT1) inhibitor. It inhibits 14C-leucine uptake and cell growth in human colon cancer-derived ...