ABT-102 - CAS 808756-71-0
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
ABT-102
Catalog Number:
808756-71-0
Synonyms:
1-[(1R)-5-tert-butyl-2,3-dihydro-1H-inden-1-yl]-3-(1H-indazol-4-yl)urea
CAS Number:
808756-71-0
Description:
ABT 102 is a selective transient receptor potential vanilloid 1 (TRPV1) receptor antagonist with IC50 values to be 5-7 nM. No recent reports of development identified for phase-I development in Pain in USA.
Molecular Weight:
348.44
Molecular Formula:
C21H24N4O
Quantity:
Milligrams-Grams
Quality Standard:
In-house standard
COA:
Inquire
MSDS:
Inquire
Canonical SMILES:
CC(C)(C)C1=CC2=C(C=C1)C(CC2)NC(=O)NC3=CC=CC4=C3C=NN4
InChI:
InChI=1S/C21H24N4O/c1-21(2,3)14-8-9-15-13(11-14)7-10-18(15)24-20(26)23-17-5-4-6-19-16(17)12-22-25-19/h4-6,8-9,11-12,18H,7,10H2,1-3H3,(H,22,25)(H2,23,24,26)/t18-/m1/s1
InChIKey:
TYOYXJNGINZFET-GOSISDBHSA-N
Targets:
TRP Channel
Current Developer:
Originator Abbott Laboratories
Chemical Structure
CAS 808756-71-0 ABT-102

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