A-438079 HCl - CAS 899431-18-6
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
A-438079 HCl
Catalog Number:
899431-18-6
CAS Number:
899431-18-6
Description:
A-438079 HCl is a potent, and selective P2X7 receptor antagonist with pIC50 of 6.9.
Molecular Weight:
342.61
Molecular Formula:
C13H10Cl3N5
COA:
Inquire
MSDS:
Inquire
Canonical SMILES:
C1=CC(=C(C(=C1)Cl)Cl)C2=NN=NN2CC3=CN=CC=C3.Cl
Targets:
P2X Receptor

Related P2X Receptor Products


CAS 309712-55-8 GW791343 HCl

GW791343 HCl
(CAS: 309712-55-8)

GW791343 HCl is aHCl salt form of GW791343, which is a non-competitive allosteric modulator of human P2X7 receptor inhibitor with pIC50 of 7.

CAS 861393-28-4 A-740003

A-740003
(CAS: 861393-28-4)

A-740003 is potent, selective and competitive P2X7 receptor antagonist. Its IC50 values are 18 and 40 nM for rat and human receptors respectively measured by ag...

CAS 475205-49-3 A-317491 sodium

A-317491 sodium
(CAS: 475205-49-3)

A-317491 is a potent and selective non-nucleotide antagonist of P2X3 and P2X2/3 receptors stimulate the pronociceptive effects of ATP upon activation.

CAS 987-65-5 ATP

ATP
(CAS: 987-65-5)

ATP is a disodium salt form of adenosine-triphosphate which is a multifunctional nucleoside triphosphate.

CAS 1019779-04-4 GW 791343 hydrochloride

GW 791343 hydrochloride
(CAS: 1019779-04-4)

The hydrochlorie salt form of GW791343 that is a non-competitive inhibitor of human P2X7 receptors amd it seems to show species-specific activity which is proba...

CAS 227088-94-0 AZ11645373

AZ11645373
(CAS: 227088-94-0)

AZ11645373 is a potent and selective human P2X7 antagonist (KB values are 5 - 7 and > 10,000 nM at hP2X7 and rP2X7 respectively) that is completely without effe...

CAS 127191-97-3 KN-62

KN-62
(CAS: 127191-97-3)

KN-62 suppresses the A23187-induced autophosphorylation of Ca2+/CaM kinase in PC12 D cells.

A-438079 HCl
(CAS: 899431-18-6)

A-438079 HCl is a potent, and selective P2X7 receptor antagonist with pIC50 of 6.9.

CAS 870061-27-1 A 839977

A 839977
(CAS: 870061-27-1)

A-839977 is a novel and selective P2X7 antagonist. It blocks BzATP-evoked calcium influx at recombinant human, rat and mouse P2X7 receptors with IC50 values 20,...

CAS 865305-30-2 AF 353

AF 353
(CAS: 865305-30-2)

AF-353 is a novel, potent and orally bioavailable P2X3/P2X2/3 receptor antagonist. It is a highly potent inhibitor of α,β-meATP-evoked intracellular calcium flu...