A 419259 trihydrochloride - CAS 1435934-25-0
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
A 419259 trihydrochloride
Catalog Number:
1435934-25-0
Synonyms:
A419259 trihydrochloride; A-419259 trihydrochloride; RK 20449 trihydrochloride; RK20449 trihydrochloride; RK-20449 trihydrochloride
CAS Number:
1435934-25-0
Description:
Potent Hck inhibitor (IC50 = 0.43 nM). Also inhibits other Src family kinases (SFKs). Suppresses proliferation and induces apoptosis in CML cell lines including CD34+. Also inhibits acute myeloid leukemia (AML) stem cell proliferation in vitro and in vivo.
Molecular Weight:
592.0
Molecular Formula:
C29H37Cl3N6O
COA:
Inquire
MSDS:
Inquire
Targets:
Src
Chemical Structure
CAS 1435934-25-0 A 419259 trihydrochloride

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CAS 1435934-25-0 A 419259 trihydrochloride

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Potent Hck inhibitor (IC50 = 0.43 nM). Also inhibits other Src family kinases (SFKs). Suppresses proliferation and induces apoptosis in CML cell lines including...