A-366 - CAS 1527503-11-2
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
A-366
Catalog Number:
1527503-11-2
Synonyms:
5'-methoxy-6'-(3-pyrrolidin-1-ylpropoxy)spiro[cyclobutane-1,3'-indole]-2'-amine A-366 CHEMBL3109630 A 366 GTPL8238 SCHEMBL17106564 BDBM50446376 ZINC95921314 AKOS024458525 CS-4644 HY-12583 B4947 5'-methoxy-6'-[3-(pyrrolidin-1-yl)propoxy]spiro[cyclobutane-1
CAS Number:
1527503-11-2
Description:
A-366 is peptide-competitive inhibitor of the G9a/GLP histone lysine methyltransferase (IC50 = 3.3 nM) and is approximately 1,000-fold selective over other methyltransferases.
Molecular Weight:
329.44
Molecular Formula:
C19H27N3O2
Quantity:
Grams-Kilos
COA:
Inquire
MSDS:
Inquire
Canonical SMILES:
COC1=C(C=C2C(=C1)C3(CCC3)C(=N2)N)OCCCN4CCCC4
InChI:
1S/C19H27N3O2/c1-23-16-12-14-15(21-18(20)19(14)6-4-7-19)13-17(16)24-11-5-10-22-8-2-3-9-22/h12-13H,2-11H2,1H3,(H2,20,21)
InChIKey:
BKCDJTRMYWSXMC-UHFFFAOYSA-N
Targets:
HMTase

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