A-317491 sodium - CAS 475205-49-3
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
A-317491 sodium
Catalog Number:
475205-49-3
Synonyms:
ABT 202; 5-[(3-phenoxyphenyl)methyl-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]benzene-1,2,4-tricarboxylic acid;
CAS Number:
475205-49-3
Description:
A-317491 is a potent and selective non-nucleotide antagonist of P2X3 and P2X2/3 receptors stimulate the pronociceptive effects of ATP upon activation.
Molecular Weight:
565.57
Molecular Formula:
C33H27NO8
Quantity:
Milligrams-Grams
Quality Standard:
Enterprise Standard
COA:
Inquire
MSDS:
Inquire
Canonical SMILES:
C1CC(C2=CC=CC=C2C1)N(CC3=CC(=CC=C3)OC4=CC=CC=C4)C(=O)C5=CC(=C(C=C5C(=O)O)C(=O)O)C(=O)O
InChI:
InChI=1S/C33H27NO8/c35-30(25-17-27(32(38)39)28(33(40)41)18-26(25)31(36)37)34(29-15-7-10-21-9-4-5-14-24(21)29)19-20-8-6-13-23(16-20)42-22-11-2-1-3-12-22/h1-6,8-9,11-14,16-18,29H,7,10,15,19H2,(H,36,37)(H,38,39)(H,40,41)/t29-/m0/s1
InChIKey:
VQGBOYBIENNKMI-LJAQVGFWSA-N
Targets:
P2X Receptor
Current Developer:
Abbott Laboratories
Chemical Structure
CAS 475205-49-3 A-317491 sodium

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