A-1210477 - CAS 1668553-26-1
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
A-1210477
Catalog Number:
1668553-26-1
Synonyms:
A 1210477; A1210477.
CAS Number:
1668553-26-1
Description:
A-1210477 is a potent and selective MCL-1 inhibitor with Ki and IC50 of 0.454 nM and 26.2 nM, respectively, >100-fold selectivity over other Bcl-2 family members.
Molecular Weight:
850.04
Molecular Formula:
C46H55N7O7S
COA:
Inquire
MSDS:
Inquire
Canonical SMILES:
O=C(C(N1CCN2CCOCC2)=C(CCCOC3=C(C=CC=C4)C4=CC=C3)C5=C1C(C6=C(COC7=CC=C(N8CCN(S(=O)(N(C)C)=O)CC8)C=C7)N(C)N=C6C)=CC=C5)O
Targets:
Bcl-2 Family

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