4-Phenyl-2-pyrrolidone-1-acetamide - CAS 77472-70-9
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
4-Phenyl-2-pyrrolidone-1-acetamide
Catalog Number:
77472-70-9
Synonyms:
2-(2-Oxo-4-phenyl-pyrrolidin-1-yl)acetamide;Carphedon;4-phenylpiracetam;2-Oxo-4-phenyl-1-pyrrolidineacetamide;2-Oxo-4-phenylpyrrolidine-1-acetamide;2-(2-keto-4-phenyl-pyrrolidin-1-yl)acetamide;Phenylpiracetam;Karfedon
CAS Number:
77472-70-9
Description:
4-Phenyl-2-pyrrolidone-1-acetamide is a GABA derivative that exhibited apparent immunocorrection properties during immunosuppression induced by cyclophosphamide. It is used as a stimulant nootropic drug which can be up to 30-60 times more potent than piracetam. It may have anti-amnesic, antidepressant, anticonvulsant, antipsychotic, anxiolytic, and memory enhancement effects. It has been evaluated for its efficacy in reducing neurological deficits related to cerebral ischemia, epilepsy, and neurobehavioral disorders. At 10-100 mg/kg in mice, it can increase locomotor and antidepressant activity in the open-field and forced swimming tests, and can enhance memory in a passive avoidance response test. It was developed in 1983 in Russia. It has been listed as a banned substance by the World Anti-Doping Agency and the International Olympic Committee because of its cognitive enhancing and general stimulant properties. It is intended for research and forensic purposes only.
Molecular Weight:
218.25
Molecular Formula:
C12H14N2O2
Quantity:
Kilogram to ton
Quality Standard:
In-house standard
COA:
Inquire
MSDS:
Inquire
Canonical SMILES:
C1C(CN(C1=O)CC(=O)N)C2=CC=CC=C2
InChI:
InChI=1S/C12H14N2O2/c13-11(15)8-14-7-10(6-12(14)16)9-4-2-1-3-5-9/h1-5,10H,6-8H2,(H2,13,15)
InChIKey:
LYONXVJRBWWGQO-UHFFFAOYSA-N
Targets:
AMPAR
Current Developer:
It has been approved the listing.
Chemical Structure
CAS 77472-70-9 4-Phenyl-2-pyrrolidone-1-acetamide

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